
TY  - JOUR
A1  - Prager, Rolf H. 
A1  - Schafer, Karl 
T1  - Potential GABA<emph tye="8">B</emph> Receptor Antagonists. X The Synthesis of Further Analogues of Baclofen, Phaclofen and Saclofen
JF  - Australian Journal of Chemistry
JO  - Aust. J. Chem.
Y1  - 1997
VL  - 50
IS  - 8
SP  - 813
EP  - 824
KW  - 
UR  - https://doi.org/10.1071/C97031 
N2  - In an attempt to obtain new compounds with binding activity at the GABAB receptor site, we report the synthesis of 3-amino-2-arylpropanoic acids, and the sulfonic, phosphonic and hydroxamic acid analogues. In addition, we report the synthesis of the isomer of phaclofen, 3-amino-1-(4-chlorophenyl)-propylphosphonic acid, and the higher homologue of baclofen, 5-amino-2-(4-chlorophenyl)pentanoic acid. 
ER  -

