The Synthesis of Some Chiral 2-Aminoalkyloxazole-5-carboxylates from Isoxazol-5(2H )-ones
Matthew Cox,
Rolf H. Prager, Carina E. Svensson and Max R. Taylor
Australian Journal of Chemistry
56(9) 897 - 901
Published: 20 August 2003
Abstract
Ethyl 5-oxo-2,5-dihydroisoxazole-4-carboxylates have been N-acylated by a number of natural and synthetic phthalimidylamino acids in the presence of carbodiimides. The N-acylated products form the corresponding 2-aminoalkyloxazole-5-carboxylates smoothly when irradiated at 300 nm in acetone.https://doi.org/10.1071/CH03053
© CSIRO 2003
